The effect of added silver nitrate on the palladium-catalyzed arylation of allyltrimethylsilanes K Karabelas, C Westerlund, A Hallberg The Journal of Organic Chemistry 50 (20), 3896-3900, 1985 | 220 | 1985 |
Synthesis of (E)-(2-arylethenyl) silanes by palladium-catalyzed arylation of vinylsilanes in the presence of silver nitrate K Karabelas, A Hallberg The Journal of Organic Chemistry 51 (26), 5286-5290, 1986 | 201 | 1986 |
Palladium/phosphinated polystyrene as a catalyst in the Heck arylation. A comparative study CM Andersson, K Karabelas, A Hallberg, C Andersson The Journal of Organic Chemistry 50 (20), 3891-3895, 1985 | 165 | 1985 |
Synthesis of 1-trimethylsilyl 1, 3-dienes by the palladium-catalyzed reaction of trimethylvinylsilane with vinyl iodides/silver nitrate or vinyl triflates K Karabelas, A Hallberg The Journal of Organic Chemistry 53 (21), 4909-4914, 1988 | 115 | 1988 |
Synthesis of hydroxyquinones and related compounds: semisquaric acids,(.+-.)-terreic acid,(.+-.)-perezone and (.+-.)-isoperezone A Enhsen, K Karabelas, JM Heerding, HW Moore The Journal of Organic Chemistry 55 (4), 1177-1185, 1990 | 93 | 1990 |
Palladium-catalysed arylation of vinyltrimethylsilane in the presence of silver nitrate K Karabelas, A Hallberg Tetrahedron letters 26 (26), 3131-3132, 1985 | 72 | 1985 |
Stereoselective palladium-catalyzed synthesis of (Z)-trimethyl (2-arylethenyl) silanes by arylation of (E)-1, 2-bis (trimethylsilyl) ethylene. Effects of added halides compared … K Karabelas, A Hallberg The Journal of Organic Chemistry 54 (7), 1773-1776, 1989 | 63 | 1989 |
A class of highly selective inhibitors bind to an active state of PI3Kγ G Gangadhara, G Dahl, T Bohnacker, R Rae, J Gunnarsson, S Blaho, ... Nature chemical biology 15 (4), 348-357, 2019 | 45 | 2019 |
Discovery of highly isoform selective orally bioavailable phosphoinositide 3-kinase (PI3K)-γ inhibitors N Pemberton, M Mogemark, S Arlbrandt, P Bold, RJ Cox, C Gardelli, ... Journal of Medicinal Chemistry 61 (12), 5435-5441, 2018 | 43 | 2018 |
Trimethylsilylmethyl-1, 4-benzoquinones. Generation and trapping of o-quinone methides K Karabelas, HW Moore Journal of the American Chemical Society 112 (13), 5372-5373, 1990 | 41 | 1990 |
Peptides with immunomodulatory effects H Bergstrand, T Eriksson, K Karabelas, M Lindvall, B Sarnstrand US Patent 6,103,697, 2000 | 36 | 2000 |
Pharmaceutically active compounds H Bergstrand, K Karabelas, P Sjö US Patent 6,271,231, 2001 | 35 | 2001 |
Protein kinase inhibitors K Karabelas, M Lepistö, P Sjö US Patent 6,346,625, 2002 | 29 | 2002 |
Targets of neutrophil influx and weaponry: therapeutic opportunities for chronic obstructive airway disease CK Mårdh, J Root, M Uddin, K Stenvall, A Malmgren, K Karabelas, ... Journal of immunology research 2017, 2017 | 28 | 2017 |
Selective non zinc binding inhibitors of MMP13 C De Savi, AD Morley, A Ting, I Nash, K Karabelas, CM Wood, M James, ... Bioorganic & medicinal chemistry letters 21 (14), 4215-4219, 2011 | 26 | 2011 |
Discovery of AZD8154, a dual PI3Kγδ inhibitor for the treatment of asthma MWD Perry, K Bjorhall, P Bold, M Brulls, U Borjesson, J Carlsson, ... Journal of Medicinal Chemistry 64 (12), 8053-8075, 2021 | 24 | 2021 |
Design and synthesis of soluble and cell-permeable PI3Kδ inhibitors for long-acting inhaled administration MWD Perry, K Björhall, B Bonn, J Carlsson, Y Chen, A Eriksson, ... Journal of Medicinal Chemistry 60 (12), 5057-5071, 2017 | 24 | 2017 |
Formation of reactive o-quinone methides from the reaction of trimethylsilyl (methyl)-substituted 1, 4-benzoquinones with nucleophiles JE Ezcurra, K Karabelas, HW Moore Tetrahedron 61 (1), 275-286, 2005 | 22 | 2005 |
Pharmaceutically active compounds K Karabelas, M Lepistö, P Sjö US Patent 6,492,406, 2002 | 18 | 2002 |
Modulation of human basophil histamine release by protein kinase C inhibitors differs with secretagogue and with inhibitor. H Bergstrand, B Lundquist, K Karabelas, P Michelsen Journal of Pharmacology and Experimental Therapeutics 260 (3), 1028-1037, 1992 | 18 | 1992 |