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Kostas Karabelas
Kostas Karabelas
Yperexo Life Science Consulting
Verified email at bioglan.se
Title
Cited by
Cited by
Year
The effect of added silver nitrate on the palladium-catalyzed arylation of allyltrimethylsilanes
K Karabelas, C Westerlund, A Hallberg
The Journal of Organic Chemistry 50 (20), 3896-3900, 1985
2201985
Synthesis of (E)-(2-arylethenyl) silanes by palladium-catalyzed arylation of vinylsilanes in the presence of silver nitrate
K Karabelas, A Hallberg
The Journal of Organic Chemistry 51 (26), 5286-5290, 1986
2011986
Palladium/phosphinated polystyrene as a catalyst in the Heck arylation. A comparative study
CM Andersson, K Karabelas, A Hallberg, C Andersson
The Journal of Organic Chemistry 50 (20), 3891-3895, 1985
1651985
Synthesis of 1-trimethylsilyl 1, 3-dienes by the palladium-catalyzed reaction of trimethylvinylsilane with vinyl iodides/silver nitrate or vinyl triflates
K Karabelas, A Hallberg
The Journal of Organic Chemistry 53 (21), 4909-4914, 1988
1151988
Synthesis of hydroxyquinones and related compounds: semisquaric acids,(.+-.)-terreic acid,(.+-.)-perezone and (.+-.)-isoperezone
A Enhsen, K Karabelas, JM Heerding, HW Moore
The Journal of Organic Chemistry 55 (4), 1177-1185, 1990
931990
Palladium-catalysed arylation of vinyltrimethylsilane in the presence of silver nitrate
K Karabelas, A Hallberg
Tetrahedron letters 26 (26), 3131-3132, 1985
721985
Stereoselective palladium-catalyzed synthesis of (Z)-trimethyl (2-arylethenyl) silanes by arylation of (E)-1, 2-bis (trimethylsilyl) ethylene. Effects of added halides compared …
K Karabelas, A Hallberg
The Journal of Organic Chemistry 54 (7), 1773-1776, 1989
631989
A class of highly selective inhibitors bind to an active state of PI3Kγ
G Gangadhara, G Dahl, T Bohnacker, R Rae, J Gunnarsson, S Blaho, ...
Nature chemical biology 15 (4), 348-357, 2019
452019
Discovery of highly isoform selective orally bioavailable phosphoinositide 3-kinase (PI3K)-γ inhibitors
N Pemberton, M Mogemark, S Arlbrandt, P Bold, RJ Cox, C Gardelli, ...
Journal of Medicinal Chemistry 61 (12), 5435-5441, 2018
432018
Trimethylsilylmethyl-1, 4-benzoquinones. Generation and trapping of o-quinone methides
K Karabelas, HW Moore
Journal of the American Chemical Society 112 (13), 5372-5373, 1990
411990
Peptides with immunomodulatory effects
H Bergstrand, T Eriksson, K Karabelas, M Lindvall, B Sarnstrand
US Patent 6,103,697, 2000
362000
Pharmaceutically active compounds
H Bergstrand, K Karabelas, P Sjö
US Patent 6,271,231, 2001
352001
Protein kinase inhibitors
K Karabelas, M Lepistö, P Sjö
US Patent 6,346,625, 2002
292002
Targets of neutrophil influx and weaponry: therapeutic opportunities for chronic obstructive airway disease
CK Mårdh, J Root, M Uddin, K Stenvall, A Malmgren, K Karabelas, ...
Journal of immunology research 2017, 2017
282017
Selective non zinc binding inhibitors of MMP13
C De Savi, AD Morley, A Ting, I Nash, K Karabelas, CM Wood, M James, ...
Bioorganic & medicinal chemistry letters 21 (14), 4215-4219, 2011
262011
Discovery of AZD8154, a dual PI3Kγδ inhibitor for the treatment of asthma
MWD Perry, K Bjorhall, P Bold, M Brulls, U Borjesson, J Carlsson, ...
Journal of Medicinal Chemistry 64 (12), 8053-8075, 2021
242021
Design and synthesis of soluble and cell-permeable PI3Kδ inhibitors for long-acting inhaled administration
MWD Perry, K Björhall, B Bonn, J Carlsson, Y Chen, A Eriksson, ...
Journal of Medicinal Chemistry 60 (12), 5057-5071, 2017
242017
Formation of reactive o-quinone methides from the reaction of trimethylsilyl (methyl)-substituted 1, 4-benzoquinones with nucleophiles
JE Ezcurra, K Karabelas, HW Moore
Tetrahedron 61 (1), 275-286, 2005
222005
Pharmaceutically active compounds
K Karabelas, M Lepistö, P Sjö
US Patent 6,492,406, 2002
182002
Modulation of human basophil histamine release by protein kinase C inhibitors differs with secretagogue and with inhibitor.
H Bergstrand, B Lundquist, K Karabelas, P Michelsen
Journal of Pharmacology and Experimental Therapeutics 260 (3), 1028-1037, 1992
181992
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